Series |
Handbook of experimental pharmacology ; v. 193. |
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Handbook of experimental pharmacology ;
v. 193.
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Subject |
Adenosine -- Receptors.
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Adenosine -- Physiological aspects.
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Purinergic P1 Receptor Antagonists.
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Pharmacokinetics.
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Receptors, Purinergic P1 -- therapeutic use.
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Alt Name |
Wilson, Constance N.
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Mustafa, S. Jamal.
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Description |
1 online resource. |
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polychrome rdacc |
Bibliography Note |
Includes bibliographical references and index. |
Note |
Print version record. |
Summary |
Since their discovery, adenosine receptors have emerged as important novel molecular targets in disease and drug discovery. These proteins play important roles in the entire spectrum of disease from inflammation to immune suppression. |
Contents |
To Adenosine Receptors as Therapeutic Targets -- A1 Adenosine Receptor Antagonists, Agonists, and Allosteric Enhancers -- Recent Developments in Adenosine A2A Receptor Ligands -- Recent Developments in A2B Adenosine Receptor Ligands -- Medicinal Chemistry of the A3 Adenosine Receptor: Agonists, Antagonists, and Receptor Engineering -- Adenosine Receptors and the Heart: Role in Regulation of Coronary Blood Flow and Cardiac Electrophysiology -- Adenosine Receptors and Reperfusion Injury of the Heart -- Adenosine Receptors and Inflammation -- A1 Adenosine Receptor: Role in Diabetes and Obesity -- A3 Adenosine Receptor: Pharmacology and Role in Disease -- Adenosine Receptors and Asthma -- Adenosine Receptors, Cystic Fibrosis, and Airway Hydration -- Adenosine Receptors in Wound Healing, Fibrosis and Angiogenesis -- Adenosine Receptors and Cancer -- Adenosine Receptors and the Kidney -- Adenosine Receptors and the Central Nervous System -- Adenosine Receptors and Neurological Disease: Neuroprotection and Neurodegeneration -- Adenosine A2A Receptors and Parkinson's Disease -- Adenosine Receptor Ligands and PET Imaging of the CNS. |
ISBN |
9783540896159 |
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3540896155 |
OCLC # |
437346615 |
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